From: Pharmacokinetic/Pharmacodynamic modelling of Saxagliptin and its active metabolite, 5-hydroxy Saxagliptin in rats with Type 2 Diabetes Mellitus
Analytes
Norminal
concentration (ng/mL)
Extraction recovery (n = 5) (%)
Mean
SD
RSD
SAX
15
82.58
3.41
4.13
1000
93.37
2.07
2.22
2000
92.96
2.31
2.48
5-OH SAX
3
96.18
3.18
3.30
200
91.86
2.80
3.05
400
89.27
3.90
4.37
VIL
150
92.19
1.91